Spongosorites has yielded a bis-indole alkaloid which we have named dragmacidin G. Dragmacidin G is the first in this series of compounds to have a pyrazine ring linking the two indole rings. It also has a rare N-(2-mercaptoethyl)-guanidine side chain. Dragmacidin G shows a broad spectrum of biological activity including inhibition of methicillin-resistant Staphylococcus aureus, Mycobacterium tuberculosis, Plasmodium falciparum, and a panel of pancreatic cancer cell lines.
Machine-generated and unreviewed. Identity, structure and cross-references come straight from ChEBI's and CARD's own data; no curator has signed off on this record yet.
bis-indole alkaloid with antibiotic activityARO:3007773
ARO:3007773| Molecular formula | C22H22Br2N4 |
|---|---|
| Charge | 0 |
| Average mass | 502.2 Da |
| Monoisotopic mass | 500.02112 Da |
| Source | PubChem · retrieved 2026-08-29 |
| InChIKey | GRBPIEOBAMGKFD-UHFFFAOYSA-N |
CN1CC(N(CC1C2=CNC3=C2C=CC(=C3)Br)C)C4=CNC5=C4C=CC(=C5)Br
InChI=1S/C22H22Br2N4/c1-27-11-22(18-10-26-20-8-14(24)4-6-16(18)20)28(2)12-21(27)17-9-25-19-7-13(23)3-5-15(17)19/h3-10,21-22,25-26H,11-12H2,1-2H3
| Source | Native ID | Label | Minted CURIE | Version |
|---|---|---|---|---|
| ARO | ARO:3007775 |
dragmacidin B | antibioticmech:aro-2c3e119979 |
2026-08-30 |
Seeded from data/raw/ inventories (ARO)
Re-seeded from updated data/raw/ inventories
Re-seeded from updated data/raw/ inventories